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योगदान
वार्ता
साँचा
:
Dopaminergics
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छोटा यू॰आर॰एल
प्रिंट/निर्यात
पीडीएफ़ के रूप में डाउनलोड करें
प्रिन्ट करने लायक
पठन सेटिंग्स
साइडबार पर जाएँ
छुपाएँ
मुक्त ज्ञानकोश विकिपीडिया से
दे
वा
सं
Dopaminergics
Receptor
ligands
Agonists
Adamantanes
:
Amantadine
•
Memantine
•
Rimantadine
;
Aminotetralins
:
7-OH-DPAT
•
8-OH-PBZI
•
Rotigotine
•
UH-232
;
Benzazepines
:
6-Br-APB
•
Fenoldopam
•
SKF-38,393
•
SKF-77,434
•
SKF-81,297
•
SKF-82,958
•
SKF-83,959
;
Ergolines
:
Bromocriptine
•
Cabergoline
•
Dihydroergocryptine
•
Lisuride
•
LSD
•
Pergolide
;
Dihydrexidine derivatives
:
2-OH-NPA
•
A-86,929
•
Ciladopa
•
Dihydrexidine
•
Dinapsoline
•
Dinoxyline
•
Doxanthrine
;
Others
:
A-68,930
•
A-77,636
•
A-412,997
•
ABT-670
•
ABT-724
•
Aplindore
•
Apomorphine
•
Aripiprazole
•
Bifeprunox
•
BP-897
•
CY-208,243
•
Dizocilpine
•
Etilevodopa
•
Flibanserin
•
Ketamine
•
Melevodopa
•
Modafinil
•
Pardoprunox
•
Phencyclidine
•
PD-128,907
•
PD-168,077
•
PF-219,061
•
Piribedil
•
Pramipexole
•
Propylnorapomorphine
•
Pukateine
•
Quinagolide
•
Quinelorane
•
Quinpirole
•
RDS-127
•
Ro10-5824
•
Ropinirole
•
Rotigotine
•
Roxindole
•
Salvinorin A
•
SKF-89,145
•
Sumanirole
•
Terguride
•
Umespirone
•
WAY-100,635
Antagonists
Typical antipsychotics
:
Acepromazine
•
Azaperone
•
Benperidol
•
Bromperidol
•
Clopenthixol
•
Chlorpromazine
•
Chlorprothixene
•
Droperidol
•
Flupentixol
•
Fluphenazine
•
Fluspirilene
•
Haloperidol
•
Loxapine
•
Mesoridazine
•
Methotrimeprazine
•
Nemonapride
•
Penfluridol
•
Perazine
•
Periciazine
•
Perphenazine
•
Pimozide
•
Prochlorperazine
•
Promazine
•
Sulforidazine
•
Sulpiride
•
Sultopride
•
Thioridazine
•
Thiothixene
•
Trifluoperazine
•
Triflupromazine
•
Trifluperidol
•
Zuclopenthixol
;
Atypical antipsychotics
:
Amisulpride
•
Asenapine
•
Blonanserin
•
Carpipramine
•
Clocapramine
•
Clozapine
•
Gevotroline
•
Iloperidone
•
Lurasidone
•
Melperone
•
Molindone
•
Mosapramine
•
Ocaperidone
•
Olanzapine
•
Paliperidone
•
Perospirone
•
Piquindone
•
Quetiapine
•
Remoxipride
•
Risperidone
•
Sertindole
•
Tiospirone
•
Ziprasidone
•
Zotepine
;
Antiemetics
:
AS-8112
•
Alizapride
•
Bromopride
•
Clebopride
•
Domperidone
•
Metoclopramide
•
Thiethylperazine
;
Others
:
Amoxapine
•
Buspirone
•
Butaclamol
•
Ecopipam
•
EEDQ
•
Eticlopride
•
Fananserin
•
L-745,870
•
Nafadotride
•
Nuciferine
•
PNU-99,194
•
Raclopride
•
Sarizotan
•
SB-277,011-A
•
SCH-23,390
•
SKF-83,566
•
SKF-83,959
•
Sonepiprazole
•
Spiperone
•
Spiroxatrine
•
Stepholidine
•
Tetrahydropalmatine
•
Tiapride
•
UH-232
•
Yohimbine
Reuptake inhibitors
Plasmalemmal
DAT inhibitors
Piperazines
:
DBL-583
•
GBR-12,935
•
Nefazodone
•
Vanoxerine
;
Piperidines
:
BTCP
•
Desoxypipradrol
•
Dextromethylphenidate
•
Difemetorex
•
Ethylphenidate
•
Methylnaphthidate
•
Methylphenidate
•
Phencyclidine
•
Pipradrol
;
Pyrrolidines
:
Diphenylprolinol
•
Methylenedioxypyrovalerone
(MDPV) •
Naphyrone
•
Prolintane
•
Pyrovalerone
;
Tropanes
:
β-CPPIT
•
Altropane
•
Brasofensine
•
CFT
•
Cocaine
•
Dichloropane
•
Difluoropine
•
FE-β-CPPIT
•
FP-β-CPPIT
•
Ioflupane (
123
I)
•
Iometopane
•
RTI-112
•
RTI-113
•
RTI-121
•
RTI-126
•
RTI-150
•
RTI-177
•
RTI-229
•
RTI-336
•
Tenocyclidine
•
Tesofensine
•
Troparil
•
Tropoxane
•
WF-11
•
WF-23
•
WF-31
•
WF-33
;
Others
:
Adrafinil
•
Armodafinil
•
Amfonelic acid
•
Amineptine
•
Benzatropine
(Benztropine) •
Bromantane
•
BTQ
•
BTS-74,398
•
Bupropion
(Amfebutamone) •
Ciclazindol
•
Diclofensine
•
Dimethocaine
•
Diphenylpyraline
•
Dizocilpine
•
DOV-102,677
•
DOV-21,947
•
DOV-216,303
•
Etybenzatropine
(Ethylbenztropine) •
EXP-561
•
Fencamine
•
Fencamfamine
•
Fezolamine
•
GYKI-52,895
•
Indatraline
•
Ketamine
•
Lefetamine
•
Levophacetoperane
•
LR-5182
•
Manifaxine
•
Mazindol
•
Medifoxamine
•
Mesocarb
•
Modafinil
•
Nefopam
•
Nomifensine
•
NS-2359
•
O-2172
•
Pridefrine
•
Propylamphetamine
•
Radafaxine
•
SEP-225,289
•
SEP-227,162
•
Sertraline
•
Sibutramine
•
Tametraline
•
Tripelennamine
Vesicular
VMAT
inhibitors
Deserpidine
•
Ibogaine
•
Reserpine
•
Tetrabenazine
Releasing agents
Morpholines
:
Fenbutrazate
•
Morazone
•
Phendimetrazine
•
Phenmetrazine
;
Oxazolines
:
4-Methylaminorex
(4-MAR, 4-MAX) •
Aminorex
•
Clominorex
•
Cyclazodone
•
Fenozolone
•
Fluminorex
•
Pemoline
•
Thozalinone
;
Phenethylamines
(also
amphetamines
,
cathinones
,
phentermines
, etc):
2-Hydroxyphenethylamine
(2-OH-PEA) •
4-CAB
•
4-Methylamphetamine
(4-MA) •
4-Methylmethamphetamine
(4-MMA) •
Alfetamine
•
Amfecloral
•
Amfepentorex
•
Amfepramone
•
Amphetamine
(
Dextroamphetamine
,
Levoamphetamine
) •
Amphetaminil
•
β-Methylphenethylamine
(β-Me-PEA) •
Benzodioxolylbutanamine
(BDB) •
Benzodioxolylhydroxybutanamine
(BOH) •
Benzphetamine
•
Buphedrone
•
Butylone
•
Cathine
•
Cathinone
•
Clobenzorex
•
Clortermine
•
D-Deprenyl
•
Dimethoxyamphetamine
(DMA) •
Dimethoxymethamphetamine
(DMMA) •
Dimethylamphetamine
•
Dimethylcathinone
(Dimethylpropion, metamfepramone) •
Ethcathinone
(Ethylpropion) •
Ethylamphetamine
•
Ethylbenzodioxolylbutanamine
(EBDB) •
Ethylone
•
Famprofazone
•
Fenethylline
•
Fenproporex
•
Flephedrone
•
Fludorex
•
Furfenorex
•
Hordenine
•
Lophophine
(Homomyristicylamine) •
Mefenorex
•
Mephedrone
•
Methamphetamine
(Desoxyephedrine, Methedrine;
Dextromethamphetamine
,
Levomethamphetamine
) •
Methcathinone
(Methylpropion) •
Methedrone
•
Methoxymethylenedioxyamphetamine
(MMDA) •
Methoxymethylenedioxymethamphetamine
(MMDMA) •
Methylbenzodioxolylbutanamine
(MBDB) •
Methylenedioxyamphetamine
(MDA, tenamfetamine) •
Methylenedioxyethylamphetamine
(MDEA) •
Methylenedioxyhydroxyamphetamine
(MDOH) •
Methylenedioxymethamphetamine
(MDMA) •
Methylenedioxymethylphenethylamine
(MDMPEA, homarylamine) •
Methylenedioxyphenethylamine
(MDPEA, homopiperonylamine) •
Methylone
•
Ortetamine
•
Parabromoamphetamine
(PBA) •
Parachloroamphetamine
(PCA) •
Parafluoroamphetamine
(PFA) •
Parafluoromethamphetamine
(PFMA) •
Parahydroxyamphetamine
(PHA) •
Paraiodoamphetamine
(PIA) •
Paredrine
(Norpholedrine, Oxamphetamine) •
Phenethylamine
(PEA) •
Pholedrine
•
Phenpromethamine
•
Prenylamine
•
Propylamphetamine
•
Tiflorex
(Flutiorex) •
Tyramine
(TRA) •
Xylopropamine
•
Zylofuramine
;
Piperazines
:
2,5-Dimethoxy-4-bromobenzylpiperazine
(2C-B-BZP) •
Benzylpiperazine
(BZP) •
Methoxyphenylpiperazine
(MeOPP, paraperazine) •
Methylbenzylpiperazine
(MBZP) •
Methylenedioxybenzylpiperazine
(MDBZP, piperonylpiperazine);
Others
:
2-Amino-1,2-dihydronaphthalene
(2-ADN) •
2-Aminoindane
(2-AI) •
2-Aminotetralin
(2-AT) •
4-Benzylpiperidine
(4-BP) •
5-IAI
•
Clofenciclan
•
Cyclopentamine
•
Cypenamine
•
Cyprodenate
•
Feprosidnine
•
Gilutensin
•
Heptaminol
•
Hexacyclonate
•
Indanylaminopropane
(IAP) •
Indanorex
•
Isometheptene
•
Methylhexanamine
•
Naphthylaminopropane
(NAP) •
Octodrine
•
Phthalimidopropiophenone
•
Propylhexedrine
(
Levopropylhexedrine
) •
Tuaminoheptane
(Tuamine)
Enzyme inhibitors
Anabolism
PAH
inhibitors
3,4-Dihydroxystyrene
TH
inhibitors
3-Iodotyrosine
•
Aquayamycin
•
Bulbocapnine
•
Metirosine
•
Oudenone
AAAD
/
DDC
inhibitors
Benserazide
•
Carbidopa
•
Genistein
•
Methyldopa
Catabolism
MAO inhibitors
Nonselective
:
Benmoxin
•
Caroxazone
•
Echinopsidine
•
Furazolidone
•
Hydralazine
•
Indantadol
•
Iproclozide
•
Iproniazid
•
Isocarboxazid
•
Isoniazid
•
Linezolid
•
Mebanazine
•
Metfendrazine
•
Nialamide
•
Octamoxin
•
Paraxazone
•
Phenelzine
•
Pheniprazine
•
Phenoxypropazine
•
Pivalylbenzhydrazine
•
Procarbazine
•
Safrazine
•
Tranylcypromine
;
MAO-A selective
:
Amiflamine
•
Bazinaprine
•
Befloxatone
•
Befol
•
Brofaromine
•
Cimoxatone
•
Clorgiline
•
Esuprone
•
Harmala alkaloids
(
Harmine
,
Harmaline
,
Tetrahydroharmine
,
Harman
,
Norharman
, etc) •
Methylene Blue
•
Metralindole
•
Minaprine
•
Moclobemide
•
Pirlindole
•
Sercloremine
•
Tetrindole
•
Toloxatone
•
Tyrima
;
MAO-B selective
:
D-Deprenyl
•
L-Deprenyl
(Selegiline) •
Ladostigil
•
Lazabemide
•
Milacemide
•
Mofegiline
•
Pargyline
•
Rasagiline
COMT inhibitors
Entacapone
•
Tolcapone
DBH
inhibitors
Bupicomide
•
Disulfiram
•
Dopastin
•
Fusaric acid
•
Nepicastat
•
Phenopicolinic acid
•
Tropolone
Others
Precursors
L-Phenylalanine
→
L-Tyrosine
→
L-DOPA
(Levodopa)
Cofactors
Ferrous
Iron
(Fe
2+
) •
Tetrahydrobiopterin
•
Vitamin B
3
(
Niacin
,
Nicotinamide
→
NADPH
) •
Vitamin B
6
(
Pyridoxine
,
Pyridoxamine
,
Pyridoxal
→
Pyridoxal Phosphate
) •
Vitamin B
9
(
Folic acid
→
Tetrahydrofolic acid
) •
Vitamin C
(
Ascorbic acid
) •
Zinc
(Zn
2+
)
Others
Activity Enhancers
:
Benzofuranylpropylaminopentane
(BPAP) •
Phenylpropylaminopentane
(PPAP);
Toxins
:
Oxidopamine
(6-Hydroxydopamine)
श्रेणी
:
Drug templates by receptor, channel, or pump
छुपी हुई श्रेणियाँ:
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